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2427041
glucopeptidos
Description
tarea farmacología especial Mind Map on glucopeptidos, created by jelramirezav on 03/04/2015.
No tags specified
farmacología especial
tarea
Mind Map by
jelramirezav
, updated more than 1 year ago
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Created by
jelramirezav
over 9 years ago
121
1
0
Resource summary
glucopeptidos
vancomicina y teiclopanina
mec de accion
inhibe sintesis de pared celular, paso previo al de B-lactamicos
altera permeabilidad en la membrana
impide sintesis de ARN
impide union a capa de peptidoglicano
bactericida
generalidades
resistencia
sintesis de proteinas que impiden la union de la vancomicina a la unidad precursora
espectro
mas para gram +
farmacocinetica
vancomicina no se absorbe por VO
IV unica via
alcanza concentraciones liquidos asciticos, pericardicos, pleural y sinovial
via orina
resto via hepatica y biliar
inalterada
vancomicina
pilas administracion rapida
infusion lenta
60 min
aplicaciones terapeuticas
vancomicina primera eleccioncontra s. aureus
resistente ameticilina, penicilinas, isoxasolicas y cefalosporinas de 1 generacion
infecciones por epidermidis
poco sensible a las penicilinas, isoxazolicas y a la meticilina
eleccion a pacientes alergicos a las penicilinas aureus y epidermidis
alternativa en endocarditis estreptococica
meningitis
RAMs
neurotoxicidad
neurotoxicidad del nervio acustico
perdidad de la audicon
reacciones de hipersensibilidad
trombocitopenia
disfuncion hepatica
interacciones
vancomicina incompatible en solucion
cloranfenicol, corticoesteroides, meticilina y heparina
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